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Hydroxylases
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View larger Osilodrostat
AT4277
CAS 928134-65-0
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Data sheet
| Molecular Formula | C13H10FN3 |
| Molecular Weight | 227.24 |
| CAS Numbers | 928134-65-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Fc1cc(ccc1[C@H]1CCc2cncn12)C#N |
| References | Li L, et al. Osilodrostat [LCI699], a potent 11?-hydroxylase inhibitor, administered in combination with the multireceptor-targeted somatostatin analog pasireotide A 13-week study in rats. Toxicol Appl Pharmacol. 2015 Aug 1;286[3] 224-33. |
More info
Osilodrostat (LCI699) (LCI699) is an effective inhibitor of human 11?-hydroxylase (IC50: 2.5 nM) and aldosterone synthase (IC50: 0.7 nM).