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View larger CB2RFAAH modulator-3
AT67747
CAS 2876918-67-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Data sheet
| Molecular Formula | C22H31NO2 |
| Molecular Weight | 341.49 |
| CAS Numbers | 2876918-67-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCCCOc1ccccc1C(=O)NC12CC3CC(CC(C3)C1)C2 |
| References | Francesca Intranuovo, et al. Development of N-[1-Adamantyl]benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. J Med Chem. 2023 Jan 12;66[1] 235-250. |
More info
CB2RFAAH modulator-3 (compound 27) is a modulator targeting CB2R and FAAH, acting as a CB2R agonist with a Ki value of 20.1 nM and a CB1R agonist with a Ki value of 67.6 nM, while inhibiting FAAH with an IC50 value of 3.4 ?M. This compound has research value in cancer, neurodegenerative disease-related inflammatory cascades, and COVID-19 infection.