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View larger Org 25543 hydrochloride
AT22126
CAS 495076-64-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $36.90 | Total: $3,690.00 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 5 | $69.70 | Total: $348.50 |
Data sheet
| Molecular Formula | C24H33ClN2O4 |
| Molecular Weight | 448.983 |
| CAS Numbers | 495076-64-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.COc1cc(cc(OC)c1OCc1ccccc1)C(=O)NCC1(CCCC1)N(C)C |
| References | W L Caulfield, et al.The first potent and selective inhibitors of the glycine transporter type 2.J Med Chem . 2001 Aug 16;44[17] 2679-82. |
More info
Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2). Displays no activity at GlyT1 or 56 other common biological targets (? 100 ?M), in a glycine uptake assay in CHO cells.