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Kinase Inhibitors
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View larger (EZ)-BIX02188
AT6324
CAS 1094614-84-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Data sheet
| Molecular Formula | C25H24N4O2 |
| Molecular Weight | 412.48 |
| CAS Numbers | 1094614-84-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)Cc1cccc(NC(=C2C(=O)Nc3cc(ccc23)C(N)=O)c2ccccc2)c1 |
| References | Tatake RJ, et al. Biochem Biophys Res Commun, 2008, 377[1], 120-125. |
More info
BIX02188 is a specific MEK5 inhibitor (IC50: 4.3 nM), also inhibits ERK5 catalytic activity (IC50: 810 nM), and does not inhibit closely related kinases MEK12, JNK2, and ERK2.