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View larger Atuveciclib Racemate
AT10464L
CAS 1414943-88-6
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $58.65 | Total: $293.25 |
| 1 | 10 | $49.68 | Total: $496.80 |
| 1 | 25 | $42.09 | Total: $1,052.25 |
| 1 | 50 | $35.88 | Total: $1,794.00 |
| 1 | 100 | $31.05 | Total: $3,105.00 |
Data sheet
| Molecular Formula | C18H18FN5O2S |
| Molecular Weight | 387.43 |
| CAS Numbers | 1414943-88-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(F)ccc1-c1ncnc(Nc2cccc(CS(C)(=N)=O)c2)n1 |
| References | Scholz A, et al. BAY 1143572, a first-in-class, highly selective, potent and orally available inhibitor of PTEFbCDK9 currently in Phase I, shows convincing anti-tumor activity in preclinical models of acute myeloid leukemia [AML]. [abstract]. In Proceedings of the 107th Annual Meeting of the American Association for Cancer Research; 2016 Apr 16-20; New Orleans, LA. Philadelphia [PA] AACR; Cancer Res 2016;76[14 Suppl] Abstract nr 3022. |
More info
Atuveciclib Racemate (BAY-1143572 Racemate) is a racemate mixture of Atuveciclib, a potent and highly selective oral P-TEFbCDK9 inhibitor that suppresses CDK9CycT1 with an IC50 of 13 nM.