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View larger Cot inhibitor-1 hydrochloride
AT10865L
CAS
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $91.80 | Total: $459.00 |
| 1 | 10 | $77.76 | Total: $777.60 |
| 1 | 25 | $65.88 | Total: $1,647.00 |
| 1 | 50 | $56.16 | Total: $2,808.00 |
| 1 | 100 | $48.60 | Total: $4,860.00 |
Data sheet
| Molecular Formula | C27H28Cl3FN8 |
| Molecular Weight | 589.92 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N#CC1=CN=C2C(Cl)=CC(NCC3=CN(CCN4CCCCCC4)N=N3)=CC2=C1NC5=CC=C(C(Cl)=C5)F.Cl |
| References | Junjun Wu, et al. Selective inhibitors of tumor progression loci-2 [Tpl2] kinase with potent inhibition of TNF-alpha production in human whole blood. Bioorg Med Chem Lett. 2009 Jul 1;19[13] 3485-8. |
More info
Cot inhibitor-1 hydrochloride is an inhibitor of tumor progression loci-2 kinase (IC50 = 28 nM) and inhibits the production of TNF-? in human whole blood (IC50 = 5.7 nM).