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Kinase Inhibitors
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View larger Fadraciclib
ATQ0053
CAS 1070790-89-4
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $49.30 | Total: $246.50 |
| 1 | 10 | $41.76 | Total: $417.60 |
| 1 | 25 | $35.38 | Total: $884.50 |
| 1 | 50 | $30.16 | Total: $1,508.00 |
| 1 | 100 | $26.10 | Total: $2,610.00 |
Data sheet
| Molecular Formula | C21H31N7O |
| Molecular Weight | 397.52 |
| CAS Numbers | 1070790-89-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC[C@H](Nc1nc(NCc2cnc(C)cc2C)c2ncn(C(C)C)c2n1)[C@@H](C)O |
| References | Cocco E, et al. Dual CCNE1PIK3CA targeting is synergistic in CCNE1-amplifiedPIK3CA-mutated uterine serous carcinomas in vitro and in vivo. Br J Cancer. 2016 Jul 26;115[3] 303-11. |
More info
Fadraciclib (CYC065) is an orally available, second-generation ATP-competitive inhibitor of CDK2CDK9 kinases (IC50s: 526 nM).