Kinase Inhibitors

Lenacapavir View larger

Lenacapavir

AT11465

CAS 2189684-44-2

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$283.00

$283.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $127.35 Total: $12,735.00
150 $147.16 Total: $7,358.00
125 $172.63 Total: $4,315.75
110 $203.76 Total: $2,037.60
15 $240.55 Total: $1,202.75

Data sheet

Molecular FormulaC39H32ClF10N7O5S2
Molecular Weight968.28
CAS Numbers2189684-44-2
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES Code[H][C@]12C[C@@]1([H])C(F)(F)c1c2c(nn1CC(=O)N[C@@H](Cc1cc(F)cc(F)c1)c1nc(ccc1-c1ccc(Cl)c2c(NS(C)(=O)=O)nn(CC(F)(F)F)c12)C#CC(C)(C)S(C)(=O)=O)C(F)(F)F
ReferencesJohn O Link, et al. Clinical targeting of HIV capsid protein with a long-acting small molecule. Nature. 2020 Jul 1.

More info

Lenacapavir (GS-6207) is a potent capsid-targeting inhibitor of HIV replication, demonstrating anti-HIV activity with an EC50 of 100 pM in MT-4 cells.