Kinase Inhibitors

L 756423 View larger

L 756423

AT24362

CAS 216863-66-0

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$332.00

$332.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $149.40 Total: $14,940.00
150 $172.64 Total: $8,632.00
125 $202.52 Total: $5,063.00
110 $239.04 Total: $2,390.40
15 $282.20 Total: $1,411.00

Data sheet

Molecular FormulaC39H48N4O5
Molecular Weight652.82
CAS Numbers216863-66-0
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeN(C([C@H](CC1=CC=CC=C1)C[C@@H](CN2[C@H](C(NC(C)(C)C)=O)CN(CC3=CC=4C(O3)=CC=CC4)CC2)O)=O)[C@H]5C=6C(C[C@H]5O)=CC=CC6
ReferencesDorsey BD, et al. Identification of MK-944a a second clinical candidate from the hydroxylaminepentanamide isostere series of HIV protease inhibitors. J Med Chem. 2000 Sep 7;43[18] 3386-99.

More info

L 756423 (L756423) is a novel potent and selective and competitive HIV protease inhibitor with a Ki value of 0.049 nM for HIV-1 PR.L 756423 blocks the spread of HIV(IIIb)-infected MT25 lymphocytes at 0.50-0.1 nM and can be used for the study of Acquired Immunodeficiency Syndrome (AIDS).