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> Pathway Inhibitors>Enzyme Inhibitors>Kinase Inhibitors>MLCK inhibitor peptide 18 acetate

Kinase Inhibitors

MLCK inhibitor peptide 18 acetate View larger

MLCK inhibitor peptide 18 acetate

ATP1890L1

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$40.00

$40.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $34.00 Total: $170.00
110 $28.80 Total: $288.00
125 $24.40 Total: $610.00
150 $20.80 Total: $1,040.00
1100 $18.00 Total: $1,800.00

Data sheet

Molecular FormulaC62H109N23O13
Molecular Weight1384.67
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC1=CC(=CC=C1C[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC2=CC=C(C=C2)O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCN=C(N)N)N)O.CC(=O)O
ReferencesLukas et al [1999] Identification of novel classes of protein kinase inhibitors using combinatorial peptide chemistry based on functional genomics knowledge. J.Med.Chem. 42 910 PMID

More info

MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA. Cell permeable.