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Kinase Inhibitors
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View larger Ertiprotafib
AT15243
CAS 251303-04-5
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $66.30 | Total: $331.50 |
| 1 | 10 | $56.16 | Total: $561.60 |
| 1 | 25 | $47.58 | Total: $1,189.50 |
| 1 | 50 | $40.56 | Total: $2,028.00 |
| 1 | 100 | $35.10 | Total: $3,510.00 |
Data sheet
| Molecular Formula | C31H27BrO3S |
| Molecular Weight | 559.51 |
| CAS Numbers | 251303-04-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC=1C2=C(C=3C(C(Br)=C2SC1C)=CC=CC3)C4=CC(C)=C(O[C@H](CC5=CC=CC=C5)C(O)=O)C(C)=C4 |
| References | Shrestha S, et al. PTP1B inhibitor Ertiprotafib is also a potent inhibitor of IkappaB kinase beta [IKK-beta]. Bioorg Med Chem Lett. 2007 May 15;17[10] 2728-30. Epub 2007 Mar 3. |
More info
Ertiprotafib (PTP 112), a selective and potent inhibitor of protein tyrosine phosphate 1B (PTP1B) and IkappaB kinase ? (IKK-?), is a novel insulin sensitizer with potential anticancer activity for the study of type 2 diabetes and breast cancer.