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Kinase Inhibitors
- Protein Control Ligand
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View larger Tenalisib
AT13119
CAS 1639417-53-0
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.95 | Total: $114.75 |
| 1 | 10 | $19.44 | Total: $194.40 |
| 1 | 25 | $16.47 | Total: $411.75 |
| 1 | 50 | $14.04 | Total: $702.00 |
| 1 | 100 | $12.15 | Total: $1,215.00 |
Data sheet
| Molecular Formula | C23H18FN5O2 |
| Molecular Weight | 415.42 |
| CAS Numbers | 1639417-53-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC[C@H](Nc1ncnc2nc[nH]c12)c1oc2ccccc2c(=O)c1-c1cccc(F)c1 |
| References | Vakkalanka S, et al. RP6530, a dual PI3K ?? inhibitor, potentiates ruxolitinib activity in the JAK2-V617F mutant erythroleukemia cell lines. [abstract]. In Proceedings of the 106th Annual Meeting of the American Association for Cancer Research; 2015 Apr 18-22; Philadelphia, PA. Philadelphia [PA] AACR; Cancer Res 2015;75[15 Suppl] Abstract nr 2704. doi 10.11581538-7445.AM2015-2704 |
More info
Tenalisib (RP6530) (RP6530) is a potent and selective inhibitor of PI3K? and PI3K?(IC50 values of 25 and 33 nM, respectively.)