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View larger Umbralisib R-enantiomer
AT13140
CAS 1532533-69-9
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $75.15 | Total: $7,515.00 |
| 1 | 50 | $86.84 | Total: $4,342.00 |
| 1 | 25 | $101.87 | Total: $2,546.75 |
| 1 | 10 | $120.24 | Total: $1,202.40 |
| 1 | 5 | $141.95 | Total: $709.75 |
Data sheet
| Molecular Formula | C31H24F3N5O3 |
| Molecular Weight | 571.55 |
| CAS Numbers | 1532533-69-9 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)Oc1ccc(cc1F)-c1nn([C@H](C)c2oc3ccc(F)cc3c(=O)c2-c2cccc(F)c2)c2ncnc(N)c12 |
| References | Michael Weiss, et al. Combination of anti-cd20 antibody and pi3 kinase selective inhibitor. WO2014071125A1. |
More info
Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against ?PI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, ?, and ?).