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Kinase Inhibitors
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View larger PI3K?-IN-1
AT12462
CAS 1911564-39-0
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $41.65 | Total: $208.25 |
| 1 | 10 | $35.28 | Total: $352.80 |
| 1 | 25 | $29.89 | Total: $747.25 |
| 1 | 50 | $25.48 | Total: $1,274.00 |
| 1 | 100 | $22.05 | Total: $2,205.00 |
Data sheet
| Molecular Formula | C22H20F3N7O2 |
| Molecular Weight | 471.44 |
| CAS Numbers | 1911564-39-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(=O)N1CCN(C(=O)C1(C)C)c1cc(ccc1C#N)-c1cc(c2c(N)ncnn12)C(F)(F)F |
| References | Liu Q, et al. Identification of a Potent, Selective, and Efficacious Phosphatidylinositol 3-Kinase ? [PI3K?] Inhibitor for the Treatment of Immunological Disorders. J Med Chem. 2017 Jun 22;60[12] 5193-5208. |
More info
PI3K?-IN-1 is an efficacious PI3K? inhibitor (IC50 of 1.7 nM).