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Kinase Inhibitors
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View larger Tilfrinib
AT17098
CAS 1600515-49-8
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Data sheet
| Molecular Formula | C17H13N3O |
| Molecular Weight | 275.3 |
| CAS Numbers | 1600515-49-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Oc1cccc(Nc2ccnc3[nH]c4ccccc4c23)c1 |
| References | Mahmoud KA, et al. Discovery of 4-anilino ?-carbolines as novel Brk inhibitors. Bioorg Med Chem Lett. 2014 Apr 15;24[8] 1948-51. |
More info
Tilfrinib is an effective and selective inhibitor of breast tumor kinase(Brk, IC50 = 3.15 nM) which displays anti-proliferative and anti-tumor activities.