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View larger Phthalazinone pyrazole
AT21981
CAS 880487-62-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $38.25 | Total: $3,825.00 |
| 1 | 50 | $44.20 | Total: $2,210.00 |
| 1 | 25 | $51.85 | Total: $1,296.25 |
| 1 | 10 | $61.20 | Total: $612.00 |
| 1 | 5 | $72.25 | Total: $361.25 |
Data sheet
| Molecular Formula | C18H15N5O |
| Molecular Weight | 317.34 |
| CAS Numbers | 880487-62-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cc(Nc2nn(-c3ccccc3)c(=O)c3ccccc23)n[nH]1 |
| References | Prime M E, Courtney S M, Brookfield F A, et al. Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of Aurora-A kinase[J]. Journal of medicinal chemistry, 2010, 54[1] 312-319. |
More info
Phthalazinone pyrazole is potent, selective, and orally bioavailable inhibitor of Aurora-A kinase. Aurora-A is overexpressed in a variety of tumor types and displays oncogenic activity.