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View larger IRAK inhibitor 1
AT5094
CAS 1042224-63-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $62.90 | Total: $314.50 |
| 1 | 10 | $53.28 | Total: $532.80 |
| 1 | 25 | $45.14 | Total: $1,128.50 |
| 1 | 50 | $38.48 | Total: $1,924.00 |
| 1 | 100 | $33.30 | Total: $3,330.00 |
Data sheet
| Molecular Formula | C17H19N5 |
| Molecular Weight | 293.37 |
| CAS Numbers | 1042224-63-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C1CC(CCN1)Nc1cccc(n1)-c1cnc2ccccn12 |
| References | Buckley GM, et al. IRAK-4 inhibitors. Part II A structure-based assessment of imidazo[1,2-a]pyridine binding. Bioorg Med Chem Lett. 2008 Jun 1;18[11] 3291-5. |
More info
IRAK inhibitor 1 is an effective IRAK-4 inhibitor (IC50: 216 nM), is poorly active against JNK-1 (IC50: 3.801 ?M) and JNK-2 (IC50>10 ?M).