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Kinase Inhibitors
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View larger ZINC194100678
AT60269
CAS 1995025-05-2
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.10 | Total: $705.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 100 | $74.70 | Total: $7,470.00 |
Data sheet
| Molecular Formula | C10H13N5O |
| Molecular Weight | 219.24 |
| CAS Numbers | 1995025-05-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C1=C2C(NN=C2)=NC=N1)C3CCOCC3 |
| References | Zhang J, et al. Design, synthesis and biological evaluation of 1H-pyrazolo [3,4-d]pyrimidine derivatives as PAK1 inhibitors that trigger apoptosis, ER stress and anti-migration effect in MDA-MB-231 cells. Eur J Med Chem. 2020;194 112220. |
More info
ZINC194100678 is an effective PAK1 inhibitor with IC50 of 8.37?M. ZINC194100678 showed strong anti-proliferation activity, with IC50 value of 40.16?M against MDA-MB-231.