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Kinase Inhibitors
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View larger GSK-1070916
AOB87380
CAS No:942918-07-2
495 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.95 | Total: $114.75 |
| 1 | 10 | $19.44 | Total: $194.40 |
| 1 | 25 | $16.47 | Total: $411.75 |
| 1 | 50 | $14.04 | Total: $702.00 |
| 1 | 100 | $12.15 | Total: $1,215.00 |
Data sheet
| Molecular Formula | C30H33N7O |
| Molecular Weight | 507.6 |
| CAS Numbers | 942918-07-2 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 99% (HPLC) |
More info
A potent, selective and ATP competitive inhibitor of Aurora B and C kinases
References:
1. N. D. Adams, et al., Discovery of GSK1070916, a Potent and Selective Inhibitor of Aurora B/C Kinase, J. Med. Chem., (2010) 53: 3973–4001
2. K. Anderson, et al, Biochemical characterization of GSK1070916, a potent and selective inhibitor of Aurora B and Aurora C kinases with an extremely long residence time, Biochem. J. (2009) 420:259–265.