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View larger PCSK9-IN-10
AT72025
CAS 368434-98-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Data sheet
| Molecular Formula | C18H23N5O4 |
| Molecular Weight | 373.41 |
| CAS Numbers | 368434-98-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COCCNc1nc2n(C)c(=O)n(C)c(=O)c2n1Cc1cccc(OC)c1 |
| References | Qiao MQ, et al. Structure-activity relationship and biological evaluation of xanthine derivatives as PCSK9 inhibitors for the treatment of atherosclerosis. Eur J Med Chem. 2023;247 115047. |
More info
PCSK9-IN-10, a potent and orally active inhibitor of Proprotein Convertase SubtilisinKexin Type 9 (PCSK9), exhibits a half-maximal inhibitory concentration (IC50) of 6.4