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View larger PI5P4Ks-IN-2
AT72032
CAS 2766854-03-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $118.15 | Total: $590.75 |
| 1 | 10 | $100.08 | Total: $1,000.80 |
| 1 | 25 | $84.79 | Total: $2,119.75 |
| 1 | 50 | $72.28 | Total: $3,614.00 |
| 1 | 100 | $62.55 | Total: $6,255.00 |
Data sheet
| Molecular Formula | C22H23N5 |
| Molecular Weight | 357.45 |
| CAS Numbers | 2766854-03-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(CC1=CC=CC=N1)C2=C3C(=NC(=N2)C4=C(C(C)C)C=CC=C4)C=CN3C |
| References | Boffey HK, et al. Development of Selective Phosphatidylinositol 5-Phosphate 4-Kinase ? Inhibitors with a Non-ATP-competitive, Allosteric Binding Mode. J Med Chem. 2022;65[4] 3359-3370. |
More info
PI5P4Ks-IN-2 is an inhibitor of the phosphatidylinositol 5-phosphate 4-kinase PI5P4K?. Targeting the PI5P4K isoforms, PI5P4Ks-IN-2 inhibited PI5P4K?, PI5P4K?, PI5P4K?, and PI5P4K?+, with IC50 values of <4.3, <4.6, 6.2, and 0.32, respectively.