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Kinase Inhibitors
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View larger PERK-IN-6
AT72053
CAS 1337532-14-5
1000 Items
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $117.30 | Total: $586.50 |
| 1 | 10 | $99.36 | Total: $993.60 |
| 1 | 25 | $84.18 | Total: $2,104.50 |
| 1 | 50 | $71.76 | Total: $3,588.00 |
| 1 | 100 | $62.10 | Total: $6,210.00 |
Data sheet
| Molecular Formula | C23H22N6O |
| Molecular Weight | 398.46 |
| CAS Numbers | 1337532-14-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC1=C2C(=CN(C)C2=NC=N1)C=3C=C4C(=CC3)N(C(CC=5N=C(C)C=CC5)=O)CC4 |
| References | Axten JM, et al. Discovery of GSK2656157 An Optimized PERK Inhibitor Selected for Preclinical Development. ACS Med Chem Lett. 2013 Aug 12;4[10] 964-8. |
More info
PERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).