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Kinase Inhibitors
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View larger BSJ-04-122
AT73182
CAS 2513289-74-0
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $25.50 | Total: $127.50 |
| 1 | 10 | $21.60 | Total: $216.00 |
| 1 | 25 | $18.30 | Total: $457.50 |
| 1 | 50 | $15.60 | Total: $780.00 |
| 1 | 100 | $13.50 | Total: $1,350.00 |
Data sheet
| Molecular Formula | C15H12ClN5O |
| Molecular Weight | 313.74 |
| CAS Numbers | 2513289-74-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C1=C2C(NC=C2Cl)=NC=N1)C3=C(NC(C=C)=O)C=CC=C3 |
| References | Jiang J, et al. Discovery of Covalent MKK47 Dual Inhibitor. Cell Chem Biol. 2020 Dec 17;27[12] 1553-1560.e8. |
More info
BSJ-04-122 is a covalent dual inhibitor of MKK4 and MKK7, demonstrating IC50 values of 4 nM and 181 nM, respectively. [BSJ-04-122] can be used for cancer research.