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Kinase Inhibitors
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View larger LY2857785
ATQ0060
CAS 1619903-54-6
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Data sheet
| Molecular Formula | C26H36N6O |
| Molecular Weight | 448.6 |
| CAS Numbers | 1619903-54-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)c1n(C)nc2ccc(cc12)-c1ccnc(N[C@H]2CC[C@@H](CC2)NC2CCOCC2)n1 |
| References | Yin T, et al. A novel CDK9 inhibitor shows potent antitumor efficacy in preclinical hematologic tumor models. Mol Cancer Ther. 2014 Jun;13[6] 1442-56. Mol Cancer Ther. 2014 Jun;13[6] 1442-56. |
More info
LY2857785 is a type I competitive and reversible ATP kinase inhibitor against CDK7CDK8CDK9 (IC50s: 246 nM16 nM11 nM).