Metabolites

Enerisant HCl View larger

Enerisant HCl

AT70489

CAS 1152749-07-9

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$79.00

$79.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $35.55 Total: $3,555.00
150 $41.08 Total: $2,054.00
125 $48.19 Total: $1,204.75
110 $56.88 Total: $568.80
15 $67.15 Total: $335.75

Data sheet

Molecular FormulaC22H31ClN4O3
Molecular Weight434.96
CAS Numbers1152749-07-9
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(=O)(C1=CN(N=C1)C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N4CCOCC4.Cl
ReferencesHino N, et al. A Novel Potent and Selective Histamine H3 Receptor Antagonist Enerisant In Vitro Profiles, In Vivo Receptor Occupancy, and Wake-Promoting and Procognitive Effects in Rodents. J Pharmacol Exp Ther. 2020;375[2] 276-285.

More info

Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins.