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Metabolites
- Protein Control Ligand
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View larger 3-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one
AT8729
CAS 1031063-36-1
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HOW TO ORDER
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $17.10 | Total: $1,710.00 |
| 1 | 50 | $19.76 | Total: $988.00 |
| 1 | 25 | $23.18 | Total: $579.50 |
| 1 | 10 | $27.36 | Total: $273.60 |
| 1 | 5 | $32.30 | Total: $161.50 |
Data sheet
| Molecular Formula | C18H13NO |
| Molecular Weight | 259.3 |
| CAS Numbers | 1031063-36-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=CC(=O)C=1C=CC=NC1)C2=CC3=C(C=C2)C=CC=C3 |
| References | Horley N J , Beresford K J M , Chawla T , et al. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones Overcoming cisplatin resistance in CYP1B1-overexpressing lines[J]. European Journal of Medicinal Chemistry, 2017, 129 159-174. |
More info
DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 nM, respectively)