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mTOR
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View larger PI3K?mTOR-IN-1
AT12589
CAS 1013098-90-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $474.30 | Total: $2,371.50 |
| 1 | 10 | $401.76 | Total: $4,017.60 |
| 1 | 25 | $340.38 | Total: $8,509.50 |
| 1 | 50 | $290.16 | Total: $14,508.00 |
| 1 | 100 | $251.10 | Total: $25,110.00 |
Data sheet
| Molecular Formula | C16H18N6O |
| Molecular Weight | 310.35 |
| CAS Numbers | 1013098-90-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1N(C=2C(C=C1C=3C=NNC3)=C(C)N=C(N)N2)C4CCCC4 |
| References | Le PT, et al. Design and synthesis of a novel pyrrolidinyl pyrido pyrimidinone derivative as a potent inhibitor of PI3K? and mTOR. Bioorg Med Chem Lett. 2012 Aug 1;22[15] 5098-103. |
More info
PI3K?mTOR-IN-1 is a potent dual inhibitor of PI3K?mTOR, with an IC50 of 7 nM for PI3K? in a cell assay and Kis of 12.5 nM and 10.6 nM for mTOR and PI3K? [in a cell-free assay], respectively.