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View larger Vofopitant dihydrochloride
AT13329L
CAS 168266-51-1
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $38.25 | Total: $3,825.00 |
| 1 | 50 | $44.20 | Total: $2,210.00 |
| 1 | 25 | $51.85 | Total: $1,296.25 |
| 1 | 10 | $61.20 | Total: $612.00 |
| 1 | 5 | $72.25 | Total: $361.25 |
Data sheet
| Molecular Formula | C21H25Cl2F3N6O |
| Molecular Weight | 505.36 |
| CAS Numbers | 168266-51-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.COc1ccc(cc1CN[C@H]1CCCN[C@H]1c1ccccc1)-n1nnnc1C(F)(F)F |
| References | Gardner CJ, et al. GR205171 a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. Regul Pept. 1996 Aug 27;65[1] 45-53. |
More info
Vofopitant dihydrochloride (GR 205171A) is an orally available, selective tachykinin NK1 receptor antagonist that inhibits [3H]SP binding to NK1 with pKi values of 9.5 and 10.6, respectively. It is a potential compound for the treatment of pathological vomiting.