> G Protein-Coupled Receptor Ligands>Neuropeptide Receptors>M 1145 acetate

Neuropeptide Receptors

M 1145 acetate View larger

M 1145 acetate

ATP1991L

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$526.00

$526.00 per mg

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Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $236.70 Total: $23,670.00
150 $273.52 Total: $13,676.00
125 $320.86 Total: $8,021.50
110 $378.72 Total: $3,787.20
15 $447.10 Total: $2,235.50

Data sheet

Molecular FormulaC130H209N37O34
Molecular Weight2834.28
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(O)=O.C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@H](C)NC([C@H](CC(C)C)NC([C@H](C)NC([C@H]1N(C([C@H]2N(C([C@H]3N(C([C@H](CC(C)C)NC([C@H](C(C)C)NC([C@H]4N(C(CNC([C@H](CC(C)C)NC([C@H](CC(C)C)NC([C@H](CC5=CC=C(O)C=C5)NC(CNC([C@H](C)NC([C@H](CO)NC([C@H](CC(N)=O)NC([C@H](CC(C)C)NC([C@H]([C@H](O)C)NC([C@H](CC6=CNC7=C6C=CC=C7)NC([C@H](CC(N)=O)NC(CNC([C@H](CCCNC(N)=N)NC(CNC([C@H](CCCNC(N)=N)N)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)CCC4)=O)=O)=O)CCC3)=O)CCC2)=O)CCC1)=O)=O)=O)=O)=O
ReferencesRunesson J, Saar I, Lundstr

More info

M1145 acetate, a chimeric peptide, is a selective galanin receptor type 2 (GAL2) agonist, with a Ki of 6.55 nM. M1145 acetate shows more than 90-fold higher affinity for GAL2 over GAL1 (Ki=587 nM) and a 76-fold higher affinity over GalR3 (Ki=497 nM). M1145 acetate has an additive effect on the signal transduction of galanin[1].