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> G Protein-Coupled Receptor Ligands>Neuropeptide Receptors>M617 acetate

Neuropeptide Receptors

M617 acetate View larger

M617 acetate

ATP1993L

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$404.00

$404.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $343.40 Total: $1,717.00
110 $290.88 Total: $2,908.80
125 $246.44 Total: $6,161.00
150 $210.08 Total: $10,504.00
1100 $181.80 Total: $18,180.00

Data sheet

Molecular FormulaC112H161N29O28
Molecular Weight2361.65
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(C)C[C@@H](C(NCC(N(CCC1)[C@@H]1C(N[C@@H](CCC(N)=O)C(N(CCC1)[C@@H]1C(N(CCC1)[C@@H]1C(NCC(N[C@@H](Cc1ccccc1)C(N[C@@H](CO)C(N(CCC1)[C@@H]1C(N[C@@H](Cc1ccccc1)C(N[C@@H](CCCNC(N)=N)C(N)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)NC([C@H](CC(C)C)NC([C@H](Cc(cc1)ccc1O)NC(CNC([C@H](C)NC([C@H](CO)NC([C@H](CC(N)=O)NC([C@H](CC(C)C)NC([C@H]([C@@H](C)O)NC([C@H](Cc1c[nH]c2c1cccc2)NC(CN)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O
ReferencesFang P, et al. Central injection of GalR1 agonist M617 facilitates GLUT4 expression in cardiac muscle of type 2 diabetic rats. Exp Gerontol. 2015;65 85-89.

More info

M617 acetate is a selective agonist of galanin receptor 1 (GAL1). M617 acetate acts through central GAL1, promotes GLUT4 expression, and enhances GLUT4 content in the cardiac muscle of type 2 diabetic rats. The Ki values are 0.23 and 5.71 nM for GAL1 and GAL2, respectively.