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View larger Compound 401
AT3586
CAS 168425-64-7
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Data sheet
| Molecular Formula | C16H15N3O2 |
| Molecular Weight | 281.31 |
| CAS Numbers | 168425-64-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=c1cc(nc2c3ccccc3ccn12)N1CCOCC1 |
| References | Ballou LM,et al. Inhibition of mammalian target of rapamycin signaling by 2-[morpholin-1-yl]pyrimido[2,1-alpha]isoquinolin-4-one. J Biol Chem. 2007 Aug 17;282[33] 24463-70. Epub 2007 Jun 11. |
More info
Compound 401 (2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one) is a synthetic DNA-PK inhibitor (IC50 = 0.28 ?M) that also targets mTOR but not PI3K.