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> Pathway Inhibitors>Enzyme Inhibitors>Peptidase>Teneligliptin HBr

Peptidase

Teneligliptin HBr View larger

Teneligliptin HBr

AOB19095

CAS 906093-29-6

Chemical Name: [(2S,4S)-4-[4-(5-Methyl-2-phenylpyrazol-3-yl)piperazin-1-yl]pyrrolidin-2-yl]-(1,3-thiazolidin-3-yl)methanone Hydrobromide

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Data sheet

Molecular FormulaC44H67N12O3S2
Molecular Weight1275.74
CAS Numbers906093-29-6
Storage Condition0°C (short term), -20°C (long term), desiccated
SolubilityDMSO
Purity98% by HPLC
SynonymTeneligliptin Hydrobromide
IUPAC/Chemical Name[(2S,4S)-4-[4-(5-Methyl-2-phenylpyrazol-3-yl)piperazin-1-yl]pyrrolidin-2-yl]-(1,3-thiazolidin-3-yl)methanone Hydrobromide
SMILES CodeCC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.Br.Br.Br.Br.Br
References1) Imazu M, Nakano A, Ito S, Hamasaki T, Kitakaze M; TOPLEVEL investigators and study coordinators. Effects of Teneligliptin on the Progressive Left Ventricular Diastolic Dysfunction in Patients with Type 2 Diabetes Mellitus in Open-Label, Marker-Stratified Randomized, Parallel-Group Comparison, Standard Treatment-Controlled Multicenter Trial (TOPLEVEL Study): Rationale and Study Design. Cardiovasc Drugs Ther. 2019 Mar 9. doi: 10.1007/s10557-019-06871-3. [Epub ahead of print] PubMed PMID: 30850916.

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Long-acting, orally-bioavailable inhibitor of dipeptidyl peptidase-4 (DPP-4), with hypoglycemic activity.