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View larger GV-150013X
AT27503L
CAS 151386-96-8
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.95 | Total: $709.75 |
| 1 | 10 | $120.24 | Total: $1,202.40 |
| 1 | 25 | $101.87 | Total: $2,546.75 |
| 1 | 50 | $86.84 | Total: $4,342.00 |
| 1 | 100 | $75.15 | Total: $7,515.00 |
Data sheet
| Molecular Formula | C33H34N4O3 |
| Molecular Weight | 534.65 |
| CAS Numbers | 151386-96-8 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C12CC3CC(C1)CC(C2)C3)N4C=5C(N(C(=O)[C@@H](NC(NC6=CC=CC=C6)=O)C4=O)C7=CC=CC=C7)=CC=CC5 |
| References | Gabriella, Finizia, and, et al. Synthesis and evaluation of novel 1,5-Benzodiazepines as potent and selective CCK-B ligands. Effect of the substitution of the N-5 phenyl with alkyl groups[J]. Bioorganic & Medicinal Chemistry Letters, 1996. |
More info
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi= 9.02.