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> Pathway Inhibitors>Enzyme Inhibitors>Peptidase>[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate

Peptidase

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate View larger

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate

ATP1931L1

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$122.00

$122.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $103.70 Total: $518.50
110 $87.84 Total: $878.40
125 $74.42 Total: $1,860.50
150 $63.44 Total: $3,172.00
1100 $54.90 Total: $5,490.00

Data sheet

Molecular FormulaC81H113N19O14
Molecular Weight1576.91
CAS Numbers3
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=CNC5=C4C=CC=C5)NC([C@H](CCC(N)=O)NC([C@@H](CC6=CC=CC=C6)NC([C@H]7N(C([C@H](CCCCN)NC([C@H]8N(C([C@@H](CCCNC(N)=N)N)=O)CCC8)=O)=O)CCC7)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
ReferencesHolst et al [2003] High constitutive signaling of the ghrelin receptor - identification of a potent inverse agonist. Mol.Endocrinol. 17 2201 PMID

More info

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.