Prostanoid Receptors

EP4 receptor antagonist 1 View larger

EP4 receptor antagonist 1

AT11211

CAS 2287259-07-6

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$91.00

$91.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $40.95 Total: $4,095.00
150 $47.32 Total: $2,366.00
125 $55.51 Total: $1,387.75
110 $65.52 Total: $655.20
15 $77.35 Total: $386.75

Data sheet

Molecular FormulaC23H21F3N4O3
Molecular Weight458.43
CAS Numbers2287259-07-6
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC=Cc1nnn(Cc2ccc(cc2)C(F)(F)F)c1C(=O)N[C@@H](C)c1ccc(cc1)C(O)=O
ReferencesYang JJ,

More info

EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 ?M) against human EP1, EP2, and EP3 receptors.