Protease

SCH79797 dihydrochloride View larger

SCH79797 dihydrochloride

AT12870

CAS 1216720-69-2

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$46.00

$46.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $20.70 Total: $2,070.00
150 $23.92 Total: $1,196.00
125 $28.06 Total: $701.50
110 $33.12 Total: $331.20
15 $39.10 Total: $195.50

Data sheet

Molecular FormulaC23H27Cl2N5
Molecular Weight444.4
CAS Numbers1216720-69-2
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCl.Cl.CC(C)c1ccc(Cn2ccc3c2ccc2nc(NC4CC4)nc(N)c32)cc1
ReferencesDi Serio C, et al. Protease-activated receptor 1-selective antagonist SCH79797 inhibits cell proliferation and induces apoptosis by a protease-activated receptor 1-independent mechanism. Basic Clin Pharmacol Toxicol. 2007 Jul;101[1] 63-9.

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SCH79797 dihydrochloride is an effective and selective antagonist of protease activated receptor 1 (PAR1) with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihydrochloride has antiproliferative and pro-apoptotic effects.