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View larger (1R,2R)-2-PCCA hydrochloride
AT13423
CAS 1609563-71-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $52.70 | Total: $263.50 |
| 1 | 10 | $44.64 | Total: $446.40 |
| 1 | 25 | $37.82 | Total: $945.50 |
| 1 | 50 | $32.24 | Total: $1,612.00 |
| 1 | 100 | $27.90 | Total: $2,790.00 |
Data sheet
| Molecular Formula | C30H39Cl2N3O |
| Molecular Weight | 528.56 |
| CAS Numbers | 1609563-71-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.CCCc1ccc(cc1)-c1ccc(cc1)N(C[C@@H](N)[C@@H](C)CC)C(=O)[C@@H]1C[C@H]1c1ccccn1 |
| References | Jin C, et al. Effect of Substitution on the Aniline Moiety of the GPR88 Agonist 2-PCCA Synthesis, Structure-Activity Relationships, and Molecular Modeling Studies. ACS Chem Neurosci. 2016 Oct 19;7[10] 1418-1432. |
More info
(1R,2R)-2-PCCA hydrochloride is a potent, selective, and blood-brain-barrier-crossing GPR88 receptor agonist with an EC50 value of 1140 n in striatal membranes of WT mice; it can be used to study the central nervous system.