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Rare Chemicals
- Protein Control Ligand
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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $134.10 | Total: $13,410.00 |
| 1 | 50 | $154.96 | Total: $7,748.00 |
| 1 | 25 | $181.78 | Total: $4,544.50 |
| 1 | 10 | $214.56 | Total: $2,145.60 |
| 1 | 5 | $253.30 | Total: $1,266.50 |
Data sheet
| Molecular Formula | C19H21N5O6S |
| Molecular Weight | 447.46 |
| CAS Numbers | 1286279-90-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1C2=C(NC(CCCC3=CC(C(N[C@@H](CCC(O)=O)C(O)=O)=O)=CS3)=C2)NC(N)=N1 |
| References | Wang L, et al. 6-Substituted Pyrrolo[2,3-d]pyrimidine Thienoyl Regioisomers as Targeted Antifolates for Folate Receptor ? and the Proton-Coupled Folate Transporter in Human Tumors. J Med Chem. 2015 Sep 10;58[17] 6938-59. |
More info
Antifolate C2 (AGF 154) has antitumor activity with an IC of 0.14 nM measured in a growth inhibition assay of human tumor cells.Antifolate C2 can be used for the study of cancer and autoimmune diseases.