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> Rare Chemicals>Bisubstrate Inhibitor 78 HCl

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Bisubstrate Inhibitor 78 HCl View larger

Bisubstrate Inhibitor 78 HCl

AT36802L

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$166.00

$166.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $141.10 Total: $705.50
110 $119.52 Total: $1,195.20
125 $101.26 Total: $2,531.50
150 $86.32 Total: $4,316.00
1100 $74.70 Total: $7,470.00

Data sheet

Molecular FormulaC25H30ClN7O5
Molecular Weight544
CAS Numbers917909-71-8
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO[C@H]1[C@@H](O[C@@H]([C@H]1O)CN(CC[C@H](N)C(O)=O)CC2=CC3=C(C=CC=C3)C=C2)N4C5=NC=NC(N)=C5N=C4.Cl
ReferencesGao Y,et al. Bisubstrate Inhibitors of Nicotinamide N-Methyltransferase [NNMT] with Enhanced Activity. J Med Chem. 2019 Jul 25;62[14] 6597-6614.

More info

Bisubstrate Inhibitor 78 HCl is an NNMT inhibitor (IC50 = 1.41 ?M) with potential anticancer activity, inhibiting the proliferation of HSC-2 oral cancer cells at 100 ?M.