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View larger Reldesemtiv
AT16728
CAS 1345410-31-2
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $135.15 | Total: $675.75 |
| 1 | 10 | $114.48 | Total: $1,144.80 |
| 1 | 25 | $96.99 | Total: $2,424.75 |
| 1 | 50 | $82.68 | Total: $4,134.00 |
| 1 | 100 | $71.55 | Total: $7,155.00 |
Data sheet
| Molecular Formula | C19H18F2N6O |
| Molecular Weight | 384.38 |
| CAS Numbers | 1345410-31-2 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC(=O)c1ccn(c1)-c1cnc(NC[C@@]2(C[C@H](F)C2)c2ncccc2F)nc1 |
| References | Hwee DT, et al. The small-molecule fast skeletal troponin activator, CK-2127107, improves exercise tolerance in a rat model of heart failure. J Pharmacol Exp Ther. 2015 Apr;353[1] 159-68. |
More info
Reldesemtiv (CK-2127107) is a selective fast skeletal muscle troponin activator with an EC50 of 3.4 ?M, enhancing exercise performance in heart failure models.