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Rare Chemicals
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $74.70 | Total: $7,470.00 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 5 | $141.10 | Total: $705.50 |
Data sheet
| Molecular Formula | C21H18F2N6O2 |
| Molecular Weight | 424.4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC1CCN(CC1)c1nc(cc(=O)[nH]1)-c1n[nH]c2ncc(cc12)-c1c(F)cccc1F |
| References | Ferri E, et al. Activation of the IRE1 RNase through remodeling of the kinase front pocket by ATP-competitive ligands. Nature communications, 2020, 11[1] 6387. |
More info
G-9807 significantly increases the RNase activity of IRE1-KR-0P by stabilizing the active dimeric unit, which acts as a variable activator of RNase.