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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $114.30 | Total: $11,430.00 |
| 1 | 50 | $132.08 | Total: $6,604.00 |
| 1 | 25 | $154.94 | Total: $3,873.50 |
| 1 | 10 | $182.88 | Total: $1,828.80 |
| 1 | 5 | $215.90 | Total: $1,079.50 |
Data sheet
| Molecular Formula | C20H24F2N4O3 |
| Molecular Weight | 406.43 |
| CAS Numbers | 1957278-93-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@H]1CN(CCN1c1cc(F)cc(F)c1)C(=O)CC[C@]1(NC(=O)NC1=O)C1CC1 |
| References | Franck Brebion, et al. Discovery of GLPG1972S201086, a Potent, Selective, and Orally Bioavailable ADAMTS-5 Inhibitor for the Treatment of Osteoarthritis. J Med Chem. 2021 Mar 25;64[6] 2937-2952. |
More info
Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.