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Rare Chemicals
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $14.40 | Total: $1,440.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 5 | $27.20 | Total: $136.00 |
Data sheet
| Molecular Formula | C22H23N7 |
| Molecular Weight | 385.46 |
| CAS Numbers | 881046-01-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)CCCn1c(N)c(-c2nc3ccccc3[nH]2)c2nc3ccccc3nc12 |
| References | Stelma T, Leaner VD. KPNB1-mediated nuclear import is required for motility and inflammatory transcription factor activity in cervical cancer cells. Oncotarget. 2017 May 16;8[20] 32833-32847. doi 10.18632oncotarget.15834. PubMed PMID 28427184; PubMed Central PMCID PMC5464831. |
More info
INI-43, an inhibitor of Nuclear Import-43, shows a significant cytotoxic effect on various cervical and oesophageal cancer cell lines by targeting Kpn?1 and interferes with the nuclear localization of Kpn?1 and known Kpn?1 cargoes, NFAT, NF?B, AP-1 and NF