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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $19.35 | Total: $1,935.00 |
| 1 | 50 | $22.36 | Total: $1,118.00 |
| 1 | 25 | $26.23 | Total: $655.75 |
| 1 | 10 | $30.96 | Total: $309.60 |
| 1 | 5 | $36.55 | Total: $182.75 |
Data sheet
| Molecular Formula | C45H69N13O14 |
| Molecular Weight | 1016.11 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C(N(CCC1)[C@@H]1C(NCC(O)=O)=O)[C@@H](NC([C@@]([C@H](C)CC)([H])NC([C@@H](NC([C@@H](C(C)C)NC([C@@H](CCCNC(N)=N)NC([C@@H](N)CC(O)=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)=O)CC3=CNC=N3.CC(O)=O |
| References | Strachan RT, et, al. Divergent transducer-specific molecular efficacies generate biased agonism at a G protein-coupled receptor [GPCR]. J Biol Chem. 2014 May 16; 289[20] 14211-24. |
More info
TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-?arr2 fusion proteins.