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> Rare Chemicals>TRV120056 acetate

Rare Chemicals

TRV120056 acetate View larger

TRV120056 acetate

AT40508L

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$43.00

$43.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $36.55 Total: $182.75
110 $30.96 Total: $309.60
125 $26.23 Total: $655.75
150 $22.36 Total: $1,118.00
1100 $19.35 Total: $1,935.00

Data sheet

Molecular FormulaC45H69N13O14
Molecular Weight1016.11
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C(N(CCC1)[C@@H]1C(NCC(O)=O)=O)[C@@H](NC([C@@]([C@H](C)CC)([H])NC([C@@H](NC([C@@H](C(C)C)NC([C@@H](CCCNC(N)=N)NC([C@@H](N)CC(O)=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)=O)CC3=CNC=N3.CC(O)=O
ReferencesStrachan RT, et, al. Divergent transducer-specific molecular efficacies generate biased agonism at a G protein-coupled receptor [GPCR]. J Biol Chem. 2014 May 16; 289[20] 14211-24.

More info

TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-?arr2 fusion proteins.