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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $11.25 | Total: $1,125.00 |
| 1 | 50 | $13.00 | Total: $650.00 |
| 1 | 25 | $15.25 | Total: $381.25 |
| 1 | 10 | $18.00 | Total: $180.00 |
| 1 | 5 | $21.25 | Total: $106.25 |
Data sheet
| Molecular Formula | C12H18N2O |
| Molecular Weight | 206.28 |
| CAS Numbers | 339068-25-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCCc1ccc(N=CNO)c(C)c1 |
| References | Seki T, et al. Cytochrome P450 4A isoform inhibitory profile of N-hydroxy-N'-[4-butyl-2-methylphenyl]-formamidine [HET0016], a selective inhibitor of 20-HETE synthesis. Biol Pharm Bull. 2005 Sep;28[9] 1651-4. |
More info
HET0016 is a potent and selective 20-HETE synthase inhibitor (IC50s: 17.7 nM, 12.1 nM, and 20.6 nM for recombinant CYP4A1-, CYP4A2-, and CYP4A3-catalyzed 20-HETE synthesis) and a selective CYP450 inhibitor, shown to inhibit angiogenesis and tumor growth.