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View larger SCP1-IN-1
AT60077
CAS 2764615-55-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $37.40 | Total: $187.00 |
| 1 | 10 | $31.68 | Total: $316.80 |
| 1 | 25 | $26.84 | Total: $671.00 |
| 1 | 50 | $22.88 | Total: $1,144.00 |
| 1 | 100 | $19.80 | Total: $1,980.00 |
Data sheet
| Molecular Formula | C20H19F3N2O7S2 |
| Molecular Weight | 520.5 |
| CAS Numbers | 2764615-55-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | FC(F)(F)Oc1ccc(cc1)S(=O)(=O)NCCOCCNC(=O)C1=Cc2ccccc2S1(=O)=O |
| References | Medellin B, et al. Targeted Covalent Inhibition of Small CTD Phosphatase 1 to Promote the Degradation of the REST Transcription Factor in Human Cells. J Med Chem. 2022;65[1] 507-519. |
More info
SCP1-IN-1 (compound SH T-62) is a potent and selective covalent inhibitor of SCP1, promoting REST degradation and reducing transcriptional activity. In certain glioblastoma cells, elevated REST protein levels drive tumor growth. SCP1-IN-1 holds potential for researching glioblastoma driven by REST transcription activity [1].