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Rare Chemicals
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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $37.80 | Total: $3,780.00 |
| 1 | 50 | $43.68 | Total: $2,184.00 |
| 1 | 25 | $51.24 | Total: $1,281.00 |
| 1 | 10 | $60.48 | Total: $604.80 |
| 1 | 5 | $71.40 | Total: $357.00 |
Data sheet
| Molecular Formula | C25H33NO5 |
| Molecular Weight | 427.53 |
| CAS Numbers | 2143463-35-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COC(=O)c1ccc(OC)c(NC(=O)COc2ccc(cc2)C(C)(C)CC(C)(C)C)c1 |
| References | Naik R, et al. Methyl 3-[3-[4-[2,4,4-Trimethylpentan-2-yl]phenoxy]-propanamido]benzoate as a Novel and Dual Malate Dehydrogenase [MDH] 12 Inhibitor Targeting Cancer Metabolism. J Med Chem. 2017;60[20] 8631-8646. |
More info
MDH1-IN-2 (7c) is a potent MDH1 inhibitor with an IC50 of 2.27 ?M for MDH1 and 27.47 ?M for MDH2. MDH1-IN-2 has potential anticancer activity and can be used in the study of diseases related to the immune system.