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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $58.05 | Total: $5,805.00 |
| 1 | 50 | $67.08 | Total: $3,354.00 |
| 1 | 25 | $78.69 | Total: $1,967.25 |
| 1 | 10 | $92.88 | Total: $928.80 |
| 1 | 5 | $109.65 | Total: $548.25 |
Data sheet
| Molecular Formula | C26H22F3N7O2 |
| Molecular Weight | 521.49 |
| CAS Numbers | 2648986-65-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1C2=C(C=3C(N1)=CC=C(C3)C=4C=CC(OC)=NC4)N(N=N2)C5=CC(C(F)(F)F)=C(C=C5)N6CCNCC6 |
| References | Ouyang Y, et al. Discovery of 8-[6-Methoxypyridin-3-yl]-1-[4-[piperazin-1-yl]-3-[trifluoromethyl]phenyl]-1,5-dihydro-4H-[1,2,3]triazolo[4,5-c]quinolin-4-one [CQ211] as a Highly Potent and Selective RIOK2 Inhibitor. J Med Chem. 2022;65[11] 7833-7842. |
More info
CQ211 is a potent and selective RIOK2 inhibitor with a Kd of 6.1 nM, demonstrating significant proliferation inhibitory activity against various cancer cell lines in vitro.