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View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $165.75 | Total: $828.75 |
| 1 | 10 | $140.40 | Total: $1,404.00 |
| 1 | 25 | $118.95 | Total: $2,973.75 |
| 1 | 50 | $101.40 | Total: $5,070.00 |
| 1 | 100 | $87.75 | Total: $8,775.00 |
Data sheet
| Molecular Formula | C24H30Cl2N6O2S |
| Molecular Weight | 537.51 |
| CAS Numbers | 1215011-08-7 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(S(=O)(=O)C1=C(Cl)C=C(C=C1Cl)C=2C=C(N=CC2)N3CCNCC3)C=4C(CC(C)C)=NN(C)C4C |
| References | Weickert M, et al. Initial characterization and toxicology of an nmt inhibitor in development for hematologic malignancies. Blood. 2019;134 3362. |
More info
PCLX-001 is a small-molecule compound that acts as an orally active inhibitor of N-myristoyltransferase (NMT), specifically targeting NMT1 and NMT2 with IC50 values of 5 nM and 8 nM, respectively. This compound demonstrates anti-tumor effects and effectively inhibits the early signaling of B-cell receptor (BCR). Consequently, PCLX-001 is a valuable tool for researching B-cell malignancies [1] [2].