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View larger Tefludazine
AT67811
CAS 80680-06-4
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $173.40 | Total: $867.00 |
| 1 | 10 | $146.88 | Total: $1,468.80 |
| 1 | 25 | $124.44 | Total: $3,111.00 |
| 1 | 50 | $106.08 | Total: $5,304.00 |
| 1 | 100 | $91.80 | Total: $9,180.00 |
Data sheet
| Molecular Formula | C22H24F4N2O |
| Molecular Weight | 408.43 |
| CAS Numbers | 80680-06-4 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | FC(F)(C1=CC=C([C@H](C2=CC=C(C=C2)F)C[C@H]3N4CCN(CC4)CCO)C3=C1)F |
| References | Liljefors T, et al. Conformational analysis and structural comparisons of [1R,3S]-[+]- and [1S,3R]-[-]-tefludazine, [S]-[+]- and [R]-[-]-octoclothepin, and [+]-dexclamol in relation to dopamine receptor antagonism and amine-uptake inhibition. J Med Chem. 1988;31[2] 306-312. |
More info
Tefludazine, a novel neuroleptic with a benzindone structure, is a compound with good oral activity and antagonistic effects on dopamine and 5-hydroxytryptamine receptors. Tefludazine has shown potent dopamine (DA) antagonistic activity in in vitro and in vivo test models in mice, rats and dogs. Tefludazine is a therapeutic agent used to treat psychiatric disorders.